← Pipeline|Tixatapinarof

Tixatapinarof

Approved
CRG-2755
Source: Trial-derived·Trials: 4
Modality
Nanobody
MOA
AHRant
Target
CFTR
Pathway
Checkpoint
NMOSD
Development Pipeline
Preclinical
~Nov 2010
~Feb 2012
Phase 1
~May 2012
~Aug 2013
Phase 2
~Nov 2013
~Feb 2015
Phase 3
~May 2015
~Aug 2016
NDA/BLA
~Nov 2016
~Feb 2018
Approved
May 2018
Nov 2029
ApprovedCurrent
NCT04046407
2,500 pts·NMOSD
2023-012026-08·Terminated
NCT05683529
778 pts·NMOSD
2025-102029-11·Active
NCT04834005
645 pts·NMOSD
2022-012028-12·Completed
+1 more trial
5,192 total pts1 indication
CompletedCurrentUpcoming
Catalysts (4)
2026-08-225mo awayPh3 Readout· NMOSD
2027-09-281.5y awayPh3 Readout· NMOSD
2028-12-102.7y awayPh3 Readout· NMOSD
2029-11-163.6y awayPh3 Readout· NMOSD
Trial Timeline
Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
Approved
Recruit…
Approved
Complet…
Approved
Termina…
Approved
Active
Catalysts
Ph3 Readout
2026-08-22 · 5mo away
NMOSD
Ph3 Readout
2027-09-28 · 1.5y away
NMOSD
Ph3 Readout
2028-12-10 · 2.7y away
NMOSD
Ph3 Readout
2029-11-16 · 3.6y away
NMOSD
RecruitingActiveCompletedTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT04046407ApprovedNMOSDTerminated2500LiverFat
NCT05683529ApprovedNMOSDActive778Biomarker
NCT04834005ApprovedNMOSDCompleted645ACR20
NCT05871749ApprovedNMOSDRecruiting1269NT-proBNP
Competitors (10)
DrugCompanyPhaseTargetMOA
NidasacituzumabEli LillyApprovedCFTRTYK2i
DatoglumideAbbVieApprovedCFTRCAR-T CD19
AZN-5978AstraZenecaPhase 2/3GIP-RAHRant
SNY-7254SanofiPhase 2CFTRHER2
SNY-5894SanofiApprovedCFTRSTINGag
BII-5449BiogenPhase 3FXIaAHRant
SovarelsinBioMarinPhase 2CFTRJAK1/2i
FixatuximabLegend BiotechPreclinicalCFTRRAS(ON)i
ElratapinarofHalozymePhase 2C5AHRant
NidaratamabExelixisPhase 3FLT3AHRant