← Pipeline|GYR-4594

GYR-4594

Preclinical
Source: Trial-derived·Trials: 1
Modality
Small Molecule
MOA
BETi
Target
PLK4
Pathway
Cell Cycle
PsoriasisDLBCLUC
Development Pipeline
Preclinical
Nov 2024
Jan 2028
PreclinicalCurrent
NCT04993256
420 pts·DLBCL
2024-112028-01·Recruiting
420 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2028-01-161.8y awayInterim· DLBCL
Trial Timeline
2025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028
Preclinical
Recruit…
Catalysts
Interim
2028-01-16 · 1.8y away
DLBCL
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04993256PreclinicalDLBCLRecruiting420OS
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-179Johnson & JohnsonApprovedKRASG12CBETi
LLY-1592Eli LillyNDA/BLAFGFRBETi
SovarapivirAbbViePhase 2/3IL-13BETi
BAY-8733BayerPreclinicalAuroraABETi
BemanesiranBioNTechPhase 3PLK4HPK1i
BII-1564BiogenPhase 2PSMABETi
SovanaritideArgenxPhase 3TNFαBETi
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i