← Pipeline|Pexainavolisib

Pexainavolisib

Approved
BER-6978
Source: Trial-derived·Trials: 3
Modality
mAb
MOA
CDK2i
Target
BCMA
Pathway
PD-1/PD-L1
SMAFTDMM
Development Pipeline
Preclinical
~Aug 2009
~Nov 2010
Phase 1
~Feb 2011
~May 2012
Phase 2
~Aug 2012
~Nov 2013
Phase 3
~Feb 2014
~May 2015
NDA/BLA
~Aug 2015
~Nov 2016
Approved
Feb 2017
Oct 2031
ApprovedCurrent
NCT05870906
1,541 pts·MM
2017-052028-12·Not yet recruiting
NCT03011209
1,272 pts·FTD
2023-032031-10·Terminated
NCT06591864
873 pts·FTD
2017-022031-10·Completed
3,686 total pts2 indications
CompletedCurrentUpcoming
Catalysts (3)
2028-12-022.7y awayPh3 Readout· MM
2031-10-245.6y awayPh3 Readout· FTD
2031-10-285.6y awayPh3 Readout· FTD
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3Q4
Approved
Complet…
Approved
Not yet…
Approved
Termina…
Catalysts
Ph3 Readout
2028-12-02 · 2.7y away
MM
Ph3 Readout
2031-10-24 · 5.6y away
FTD
Ph3 Readout
2031-10-28 · 5.6y away
FTD
CompletedTerminatedNot yet recruiting|StartCompletionToday
Trials (3)
NCTPhaseIndicationStatusNEP
NCT05870906ApprovedMMNot yet recr...1541ORR
NCT03011209ApprovedFTDTerminated1272HbA1c
NCT06591864ApprovedFTDCompleted873MRD
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-3703PfizerPhase 1/2CDK2CDK2i
LLY-1956Eli LillyPhase 1/2BCMAFGFRi
TirafotisoranRochePhase 2CD38CDK2i
ABB-8696AbbViePhase 3BCMAAnti-Aβ
ABB-3951AbbViePhase 2/3TNFαCDK2i
AZN-6870AstraZenecaPhase 2/3EGFRCDK2i
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
TirasotorasibTakedaNDA/BLAIL-17ACDK2i
MavuglumideBayerApprovedGLP-1RCDK2i
DSN-3066Daiichi SankyoPhase 3IL-13CDK2i