← Pipeline|MRK-7986

MRK-7986

Phase 1/2
Source: Trial-derived·Trials: 2
Modality
Gene Therapy
MOA
SHP2i
Target
WRN
Pathway
Neuroinflam
Ewing SarcomaADPKD
Development Pipeline
Preclinical
~Mar 2023
~Jun 2024
Phase 1
Sep 2024
May 2031
Phase 1Current
NCT07869694
1,608 pts·ADPKD
2024-092031-05·Completed
NCT06938147
2,601 pts·Ewing Sarcoma
2024-102029-04·Terminated
4,209 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-04-263.1y awayPh2 Data· Ewing Sarcoma
2031-05-275.2y awayPh2 Data· ADPKD
Trial Timeline
Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3
P1/2
Complet…
P1/2
Termina…
Catalysts
Ph2 Data
2029-04-26 · 3.1y away
Ewing Sarcoma
Ph2 Data
2031-05-27 · 5.2y away
ADPKD
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07869694Phase 1/2ADPKDCompleted1608HAM-D
NCT06938147Phase 1/2Ewing SarcomaTerminated2601VA
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-2191PfizerNDA/BLAGLP-1RSHP2i
MRK-3745Merck & CoPhase 2WRNFXIai
ZorisotorasibAstraZenecaPhase 1WRNTYK2i
BMY-3371Bristol-Myers SquibbPhase 3WRNBTKi
DoxacageneSanofiApprovedPSMASHP2i
LisorapivirTakedaPreclinicalWRNBTKi
NirafutibatinibBayerPhase 2WRNPD-L1i
VRT-1576Vertex PharmaPhase 2/3RETSHP2i
SovafutibatinibModernaApprovedFcRnSHP2i
DaratuximabBioMarinPhase 1PRMT5SHP2i