← Pipeline|Tirasertib

Tirasertib

Phase 1/2
THI-8438
Source: Trial-derived·Trials: 1
Modality
Bispecific Ab
MOA
PD-1i
Target
BCMA
Pathway
Ferroptosis
WilmsMG
Development Pipeline
Preclinical
~Sep 2017
~Dec 2018
Phase 1
Mar 2019
Jul 2026
Phase 1Current
NCT03345831
1,507 pts·MG
2019-032026-07·Active
1,507 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-07-184mo awayPh2 Data· MG
Trial Timeline
Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3
P1/2
Active
Catalysts
Ph2 Data
2026-07-18 · 4mo away
MG
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03345831Phase 1/2MGActive1507EFS
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-1956Eli LillyPhase 1/2BCMAFGFRi
ABB-8696AbbViePhase 3BCMAAnti-Aβ
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
GSK-7987GSKPhase 3MDM2PD-1i
REG-2328RegeneronPhase 1BCMACDK2i
AdagratapinarofVertex PharmaPreclinicalBCMAJAK1i
NirabrutinibBioNTechPhase 2/3CDK2PD-1i
BGN-6990BeiGenePhase 2/3BCMAAuroraAi
BGN-3305BeiGenePhase 2BCMAAnti-Tau
CevinaritideGenmabPhase 2/3DLL3PD-1i