← Pipeline|GLP-5658

GLP-5658

Phase 2/3
Source: Trial-derived·Trials: 2
Modality
Nanobody
MOA
KRASG12Di
Target
FcRn
Pathway
STING
CSUBreast Ca
Development Pipeline
Preclinical
~Jun 2020
~Sep 2021
Phase 1
~Dec 2021
~Mar 2023
Phase 2
Jun 2023
Jan 2030
Phase 2Current
NCT08694895
213 pts·CSU
2023-06TBD·Active
NCT03244141
1,309 pts·Breast Ca
2025-102030-01·Terminated
1,522 total pts2 indications
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-10-287mo awayFast Track· CSU
2030-01-143.8y awayPh3 Readout· Breast Ca
Trial Timeline
Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030
P2/3
Active
P2/3
Termina…
Catalysts
Fast Track
2026-10-28 · 7mo away
CSU
Ph3 Readout
2030-01-14 · 3.8y away
Breast Ca
ActiveTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08694895Phase 2/3CSUActive213Biomarker
NCT03244141Phase 2/3Breast CaTerminated1309SRI-4
Competitors (10)
DrugCompanyPhaseTargetMOA
CevizanubrutinibJohnson & JohnsonPreclinicalFcRnCD47i
DoxarasimodMerck & CoNDA/BLAFGFRKRASG12Di
GelinaritideAbbViePreclinicalFcRnCFTRmod
ZanusertibAbbVieApprovedPCSK9KRASG12Di
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
IvotuximabGSKNDA/BLAGIP-RKRASG12Di
TalalemzoparlimabGilead SciencesPhase 1FcRnTNFi
SovafutibatinibModernaApprovedFcRnSHP2i
ITC-879Intra-CellularApprovedFcRnTYK2i
JAZ-8729Jazz PharmaPhase 2/3FcRnCAR-T BCMA