← Pipeline|Olpasotorasib

Olpasotorasib

Preclinical
GPC-8307
Source: Trial-derived·Trials: 2
Modality
siRNA
MOA
CAR-T BCMA
Target
C5
Pathway
Apoptosis
SCLCSLE
Development Pipeline
Preclinical
Jul 2018
Feb 2030
PreclinicalCurrent
NCT07003022
994 pts·SCLC
2020-112030-02·Recruiting
NCT07562101
600 pts·SCLC
2018-072027-06·Not yet recruiting
1,594 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2027-06-121.2y awayInterim· SCLC
2030-02-033.8y awayInterim· SCLC
Trial Timeline
Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
Preclinical
Not yet…
Preclinical
Recruit…
Catalysts
Interim
2027-06-12 · 1.2y away
SCLC
Interim
2030-02-03 · 3.8y away
SCLC
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07003022PreclinicalSCLCRecruiting994FEV1
NCT07562101PreclinicalSCLCNot yet recr...600ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
VoxacilimabPfizerPhase 2TYK2CAR-T BCMA
LLY-9749Eli LillyPhase 3C5FGFRi
LLY-1184Eli LillyNDA/BLAC5CD3xCD20
RHH-1546RochePhase 2/3C5CAR-T CD19
NVO-9087Novo NordiskPhase 1/2TauCAR-T BCMA
BAY-6035BayerPhase 1C5Anti-Aβ
FixazanubrutinibAmgenPhase 2PI3KαCAR-T BCMA
REG-8074RegeneronPhase 2/3KRASG12CCAR-T BCMA
ARG-1250ArgenxPhase 2C5GLP-1ag
ElratapinarofHalozymePhase 2C5AHRant