← Pipeline|Talasotorasib

Talasotorasib

Preclinical
EXE-2911
Source: Trial-derived·Trials: 2
Modality
ADC
MOA
CAR-T CD19
Target
APOC3
Pathway
NF-κB
SCDTTR AmyloidosisPBC
Development Pipeline
Preclinical
Jul 2019
Jul 2031
PreclinicalCurrent
NCT03045181
2,820 pts·TTR Amyloidosis
2019-072026-05·Not yet recruiting
NCT03375686
2,314 pts·TTR Amyloidosis
2021-052031-07·Active
5,134 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-05-111mo awayInterim· TTR Amyloidosis
2031-07-075.3y awayInterim· TTR Amyloidosis
Trial Timeline
Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3Q4
Preclinical
Not yet…
Preclinical
Active
Catalysts
Interim
2026-05-11 · 1mo away
TTR Amyloidosis
Interim
2031-07-07 · 5.3y away
TTR Amyloidosis
ActiveNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03045181PreclinicalTTR AmyloidosisNot yet recr...2820PANSS
NCT03375686PreclinicalTTR AmyloidosisActive2314OS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-1944PfizerNDA/BLAAPOC3HPK1i
DoxacapivasertibEli LillyPhase 3APOC3MDM2i
RHH-1546RochePhase 2/3C5CAR-T CD19
DatoglumideAbbVieApprovedCFTRCAR-T CD19
AZN-6294AstraZenecaPhase 2/3APOC3CD47i
ZanutinibBristol-Myers SquibbPhase 2/3APOC3BiTE
GIL-2259Gilead SciencesApprovedSMN2CAR-T CD19
BII-4342BiogenPhase 2/3CGRPCAR-T CD19
ALN-5628AlnylamPhase 1/2APOC3SGLT2i
INC-1582IncytePhase 1/2APOC3TROP-2 ADC