← Pipeline|Pexanesiran

Pexanesiran

Phase 1
UTH-8874
Source: Trial-derived·Trials: 2
Modality
ERT
MOA
FXIai
Target
BCMA
Pathway
Apoptosis
NB
Development Pipeline
Preclinical
~Aug 2016
~Nov 2017
Phase 1
Feb 2018
Jun 2029
Phase 1Current
NCT05879648
385 pts·NB
2021-062029-06·Completed
NCT04669754
485 pts·NB
2018-022026-02·Recruiting
870 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-02-201mo agoInterim· NB
2029-06-123.2y awayInterim· NB
Trial Timeline
2018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
P1
Recruit…
P1
Complet…
Catalysts
Interim
2026-02-20 · 1mo ago
NB
Interim
2029-06-12 · 3.2y away
NB
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05879648Phase 1NBCompleted385ACR20
NCT04669754Phase 1NBRecruiting485FEV1
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-1956Eli LillyPhase 1/2BCMAFGFRi
NVS-6360NovartisApprovedCD38FXIai
MRK-3745Merck & CoPhase 2WRNFXIai
ABB-8696AbbViePhase 3BCMAAnti-Aβ
AZN-1715AstraZenecaPhase 3AHRFXIai
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
BMY-9931Bristol-Myers SquibbPhase 1GPRC5DFXIai
NVO-7877Novo NordiskPreclinicalGPRC5DFXIai
TAK-8730TakedaPhase 2VEGFFXIai
REG-2328RegeneronPhase 1BCMACDK2i