← Pipeline|BRK-5301

BRK-5301

Preclinical
Source: Trial-derived·Trials: 1
Modality
siRNA
MOA
STINGag
Target
PCSK9
Pathway
Wnt
Cholangiocarcinoma
Development Pipeline
Preclinical
May 2021
Apr 2030
PreclinicalCurrent
NCT07331824
2,157 pts·Cholangiocarcinoma
2021-052030-04·Completed
2,157 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-04-114.0y awayInterim· Cholangiocarcinoma
Trial Timeline
Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
Preclinical
Complet…
Catalysts
Interim
2030-04-11 · 4.0y away
Cholangiocarcinoma
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07331824PreclinicalCholangiocarcinomaCompleted2157OS
Competitors (10)
DrugCompanyPhaseTargetMOA
RHH-5389RochePreclinicalRETSTINGag
ZanusertibAbbVieApprovedPCSK9KRASG12Di
SNY-5894SanofiApprovedCFTRSTINGag
SNY-4496SanofiPhase 2/3CD3STINGag
SNY-5783SanofiPhase 1/2METSTINGag
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
GIL-4361Gilead SciencesPreclinicalPCSK9STINGag
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
BMR-8377BioMarinPhase 1/2PCSK9BTKi
CapifutibatinibIncytePhase 3PCSK9BCL-2i