← Pipeline|Zenoinavolisib

Zenoinavolisib

NDA/BLA
LAB-3876
Source: Trial-derived·Trials: 1
Modality
ASO
MOA
FXIai
Target
PLK4
Pathway
Notch
Ovarian CaBladder Ca
Development Pipeline
Preclinical
~Mar 2016
~Jun 2017
Phase 1
~Sep 2017
~Dec 2018
Phase 2
~Mar 2019
~Jun 2020
Phase 3
~Sep 2020
~Dec 2021
NDA/BLA
Mar 2022
Feb 2030
NDA/BLACurrent
NCT06545091
322 pts·Ovarian Ca
2022-032030-02·Completed
322 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-02-183.9y awayPh3 Readout· Ovarian Ca
Trial Timeline
Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
NDA/BLA
Complet…
Catalysts
Ph3 Readout
2030-02-18 · 3.9y away
Ovarian Ca
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT06545091NDA/BLAOvarian CaCompleted322PFS
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-6360NovartisApprovedCD38FXIai
MRK-3745Merck & CoPhase 2WRNFXIai
AZN-1715AstraZenecaPhase 3AHRFXIai
BMY-9931Bristol-Myers SquibbPhase 1GPRC5DFXIai
NVO-7877Novo NordiskPreclinicalGPRC5DFXIai
TAK-8730TakedaPhase 2VEGFFXIai
BemanesiranBioNTechPhase 3PLK4HPK1i
SemazasiranBeiGenePhase 1PD-1FXIai
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci