← Pipeline|Sotorapivir

Sotorapivir

Approved
MRN-5810
Source: Trial-derived·Trials: 1
Modality
siRNA
MOA
TYK2i
Target
FLT3
Pathway
JAK/STAT
PNH
Development Pipeline
Preclinical
~Mar 2016
~Jun 2017
Phase 1
~Sep 2017
~Dec 2018
Phase 2
~Mar 2019
~Jun 2020
Phase 3
~Sep 2020
~Dec 2021
NDA/BLA
~Mar 2022
~Jun 2023
Approved
Sep 2023
Feb 2031
ApprovedCurrent
NCT04156931
1,445 pts·PNH
2023-092031-02·Active
1,445 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2031-02-114.9y awayPh3 Readout· PNH
Trial Timeline
Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2
Approved
Active
Catalysts
Ph3 Readout
2031-02-11 · 4.9y away
PNH
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04156931ApprovedPNHActive1445UPDRS
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-8168Johnson & JohnsonPhase 2/3FLT3GLP-1/GIP
NidasacituzumabEli LillyApprovedCFTRTYK2i
LisonaritideEli LillyPhase 3IL-13TYK2i
MRK-2473Merck & CoPhase 1/2Nectin-4TYK2i
ZorisotorasibAstraZenecaPhase 1WRNTYK2i
SNY-8628SanofiNDA/BLAB7-H3TYK2i
VoxacageneGilead SciencesPhase 2/3SOS1TYK2i
SotosacituzumabVertex PharmaPhase 1METTYK2i
OlpainavolisibModernaPhase 1MeninTYK2i
ARG-4339ArgenxPhase 2BCL-2TYK2i