← Pipeline|Zanutinib

Zanutinib

Approved
NWR-1131
Source: Trial-derived·Trials: 1
Modality
Fusion Protein
MOA
PI3Ki
Target
LAG-3
Pathway
DDR
ADHDWet AMD
Development Pipeline
Preclinical
~Nov 2017
~Feb 2019
Phase 1
~May 2019
~Aug 2020
Phase 2
~Nov 2020
~Feb 2022
Phase 3
~May 2022
~Aug 2023
NDA/BLA
~Nov 2023
~Feb 2025
Approved
May 2025
Oct 2026
ApprovedCurrent
NCT04779773
1,899 pts·ADHD
2025-052026-10·Active
1,899 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2026-10-146mo awayPh3 Readout· ADHD
Trial Timeline
Q3Q42026Q2Q3Q4
Approved
Active
Catalysts
Ph3 Readout
2026-10-14 · 6mo away
ADHD
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04779773ApprovedADHDActive1899SeizFreq
Competitors (10)
DrugCompanyPhaseTargetMOA
TiramavacamtenRochePreclinicalSGLT2PI3Ki
NVS-5126NovartisPhase 3SHP2PI3Ki
ABB-3060AbbViePhase 2LAG-3CGRPant
VoxacilimabAstraZenecaPhase 1/2GLP-1RPI3Ki
CapifutibatinibSanofiApprovedPRMT5PI3Ki
RimatenlimabNovo NordiskPhase 2/3SGLT2PI3Ki
PolazasiranAmgenPhase 2LAG-3PCSK9i
REG-3155RegeneronPhase 1/2MDM2PI3Ki
ALN-6288AlnylamApprovedLAG-3KRASG12Ci
SovarelsinAlnylamPhase 2/3LAG-3MALT1i