← Pipeline|Pexasertib

Pexasertib

Approved
NUE-7683
Source: Trial-derived·Trials: 2
Modality
Vaccine
MOA
JAK1/2i
Target
MET
Pathway
Proteasome
ADPKD
Development Pipeline
Preclinical
~Aug 2011
~Nov 2012
Phase 1
~Feb 2013
~May 2014
Phase 2
~Aug 2014
~Nov 2015
Phase 3
~Feb 2016
~May 2017
NDA/BLA
~Aug 2017
~Nov 2018
Approved
Feb 2019
Oct 2027
ApprovedCurrent
NCT04749287
1,041 pts·ADPKD
2020-11TBD·Completed
NCT05497175
1,312 pts·ADPKD
2019-022027-10·Completed
2,353 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2027-10-231.6y awayPh3 Readout· ADPKD
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
Approved
Complet…
Approved
Complet…
Catalysts
Ph3 Readout
2027-10-23 · 1.6y away
ADPKD
Completed|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04749287ApprovedADPKDCompleted1041PASI75
NCT05497175ApprovedADPKDCompleted1312Biomarker
Competitors (10)
DrugCompanyPhaseTargetMOA
FixanesiranAbbViePreclinicalRETJAK1/2i
SNY-5783SanofiPhase 1/2METSTINGag
MotavorutinibAmgenPhase 3CDK4/6JAK1/2i
SotosacituzumabVertex PharmaPhase 1METTYK2i
VRT-9481Vertex PharmaPhase 1/2MeninJAK1/2i
SovarelsinBioMarinPhase 2CFTRJAK1/2i
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
NiramavacamtenHansoh PharmaPhase 2SGLT2JAK1/2i
RVM-274Revolution MedicinesPhase 3METKIF18Ai
TalazasiranKymeraNDA/BLAMETCFTRmod