← Pipeline|Olpasertib

Olpasertib

Preclinical
APD-7291
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
CFTRmod
Target
MDM2
Pathway
STING
LNRBPAH
Development Pipeline
Preclinical
Oct 2017
Jun 2027
PreclinicalCurrent
NCT05567152
2,761 pts·LN
2023-022026-02·Recruiting
NCT04193181
1,613 pts·LN
2017-102027-06·Completed
4,374 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-02-012mo agoInterim· LN
2027-06-281.2y awayInterim· LN
Trial Timeline
Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3
Preclinical
Complet…
Preclinical
Recruit…
Catalysts
Interim
2026-02-01 · 2mo ago
LN
Interim
2027-06-28 · 1.2y away
LN
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05567152PreclinicalLNRecruiting2761OS
NCT04193181PreclinicalLNCompleted1613BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-6079Eli LillyPhase 2MDM2PRMT5i
LLY-4358Eli LillyPhase 3B7-H3CFTRmod
LLY-3251Eli LillyPhase 2MDM2BiTE
GelinaritideAbbViePreclinicalFcRnCFTRmod
GSK-7987GSKPhase 3MDM2PD-1i
AMG-2752AmgenPreclinicalMDM2WRNi
REG-3155RegeneronPhase 1/2MDM2PI3Ki
DarafutibatinibBioNTechPreclinicalPRMT5CFTRmod
ALN-8757AlnylamPreclinicalTIGITCFTRmod
SRP-1135SareptaPhase 2/3MDM2PD-L1i