← Pipeline|Lisosotorasib

Lisosotorasib

Phase 3
OCU-4991
Source: Trial-derived·Trials: 4
Modality
mRNA
MOA
BCMA ADC
Target
CFTR
Pathway
Angiogenesis
MCLPNHMelanoma
Development Pipeline
Preclinical
~Jul 2018
~Oct 2019
Phase 1
~Jan 2020
~Apr 2021
Phase 2
~Jul 2021
~Oct 2022
Phase 3
Jan 2023
Apr 2029
Phase 3Current
NCT05767418
2,192 pts·Melanoma
2025-052027-06·Active
NCT04674355
35 pts·MCL
2023-012028-03·Terminated
NCT07182564
1,786 pts·MCL
2024-032029-04·Terminated
+1 more trial
5,868 total pts2 indications
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (4)
2027-01-119mo awayPh3 Readout· Melanoma
2027-06-271.2y awayPh3 Readout· Melanoma
2028-03-081.9y awayPh3 Readout· MCL
2029-04-173.0y awayPh3 Readout· MCL
Trial Timeline
2023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2
P3
Termina…
P3
Active
P3
Termina…
P3
Active
Catalysts
Ph3 Readout
2027-01-11 · 9mo away
Melanoma
Ph3 Readout
2027-06-27 · 1.2y away
Melanoma
Ph3 Readout
2028-03-08 · 1.9y away
MCL
Ph3 Readout
2029-04-17 · 3.0y away
MCL
ActiveTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT05767418Phase 3MelanomaActive2192Mayo
NCT04674355Phase 3MCLTerminated35MRD
NCT07182564Phase 3MCLTerminated1786PANSS
NCT04164871Phase 3MelanomaActive1855Safety
Competitors (10)
DrugCompanyPhaseTargetMOA
NidasacituzumabEli LillyApprovedCFTRTYK2i
DatoglumideAbbVieApprovedCFTRCAR-T CD19
AZN-3724AstraZenecaPreclinicalPSMABCMA ADC
SNY-7254SanofiPhase 2CFTRHER2
SNY-5894SanofiApprovedCFTRSTINGag
OlpatinibGSKPreclinicalPD-L1BCMA ADC
GIL-9779Gilead SciencesPhase 1IL-17ABCMA ADC
SovarelsinBioMarinPhase 2CFTRJAK1/2i
FixatuximabLegend BiotechPreclinicalCFTRRAS(ON)i
SematenlimabSamsung BiologicsPhase 3PI3KαBCMA ADC