← Pipeline|Zoritapinarof

Zoritapinarof

Phase 1
INV-2380
Source: Trial-derived·Trials: 1
Modality
siRNA
MOA
PRMT5i
Target
SOS1
Pathway
Complement
LGSAtopic Derm
Development Pipeline
Preclinical
~Apr 2017
~Jul 2018
Phase 1
Oct 2018
Apr 2026
Phase 1Current
NCT06878254
1,412 pts·Atopic Derm
2018-102026-04·Not yet recruiting
1,412 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-04-193w awayInterim· Atopic Derm
Trial Timeline
Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2
P1
Not yet…
Catalysts
Interim
2026-04-19 · 3w away
Atopic Derm
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT06878254Phase 1Atopic DermNot yet recr...1412SRI-4
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-6079Eli LillyPhase 2MDM2PRMT5i
RHH-8550RocheApprovedBCL-2PRMT5i
RHH-682RochePhase 2FXIaPRMT5i
TerarelsinAbbViePreclinicalSOS1SOS1i
RibofutibatinibAstraZenecaPhase 2/3SOS1PCSK9i
TalainavolisibNovo NordiskPreclinicalKRASG12DPRMT5i
AMG-4531AmgenPhase 2/3KRASG12CPRMT5i
VoxacageneGilead SciencesPhase 2/3SOS1TYK2i
GIL-9142Gilead SciencesPhase 1FXIaPRMT5i
SemainavolisibGilead SciencesPhase 2PARPPRMT5i