← Pipeline|117-9336

117-9336

Phase 2/3
Source: Trial-derived·Trials: 1
Modality
Nanobody
MOA
KRASG12Di
Target
PLK4
Pathway
Wnt
Endometrial CaGastric CaThymoma
Development Pipeline
Preclinical
~Feb 2022
~May 2023
Phase 1
~Aug 2023
~Nov 2024
Phase 2
Feb 2025
Feb 2026
Phase 2Current
NCT08921223
2,321 pts·Endometrial Ca
2025-022026-02·Active
2,321 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-02-042mo agoPh3 Readout· Endometrial Ca
Trial Timeline
Q2Q3Q42026
P2/3
Active
Catalysts
Ph3 Readout
2026-02-04 · 2mo ago
Endometrial Ca
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08921223Phase 2/3Endometrial CaActive2321FEV1
Competitors (10)
DrugCompanyPhaseTargetMOA
DoxarasimodMerck & CoNDA/BLAFGFRKRASG12Di
ZanusertibAbbVieApprovedPCSK9KRASG12Di
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
IvotuximabGSKNDA/BLAGIP-RKRASG12Di
BemanesiranBioNTechPhase 3PLK4HPK1i
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i
ILM-2412IlluminaPhase 3PLK4AuroraAi
ROI-3353Roivant SciencesPhase 1/2PLK4IL-13i