← Pipeline|Tiracapivasertib

Tiracapivasertib

Phase 2
LYE-7669
Source: Trial-derived·Trials: 1
Modality
mRNA
MOA
KRASG12Ci
Target
JAK1
Pathway
Complement
SMARBPNH
Development Pipeline
Preclinical
~Oct 2020
~Jan 2022
Phase 1
~Apr 2022
~Jul 2023
Phase 2
Oct 2023
Apr 2029
Phase 2Current
NCT07412178
2,212 pts·SMA
2023-102029-04·Terminated
2,212 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-04-093.0y awayPh2 Data· SMA
Trial Timeline
Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2
P2
Termina…
Catalysts
Ph2 Data
2029-04-09 · 3.0y away
SMA
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07412178Phase 2SMATerminated2212HbA1c
Competitors (10)
DrugCompanyPhaseTargetMOA
IvorelsinEli LillyApprovedJAK1Menini
RHH-974RochePreclinicalJAK1MALT1i
LisolucimabNovartisApprovedCD20KRASG12Ci
GozelemzoparlimabMerck & CoPhase 2FXIaKRASG12Ci
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
PexazasiranSanofiPreclinicalFXIaKRASG12Ci
TerasacituzumabNovo NordiskNDA/BLAIL-23KRASG12Ci
FixatenlimabGSKPhase 1/2JAK1CDK4/6i
GIL-8529Gilead SciencesPhase 1/2JAK1EGFRi
ALN-6288AlnylamApprovedLAG-3KRASG12Ci