← Pipeline|Lisorasimod

Lisorasimod

Phase 2/3
GEN-4424
Source: Trial-derived·Trials: 2
Modality
ASO
MOA
PD-L1i
Target
EGFR
Pathway
Fibrosis
Fabry
Development Pipeline
Preclinical
~Jun 2015
~Sep 2016
Phase 1
~Dec 2016
~Mar 2018
Phase 2
Jun 2018
Aug 2030
Phase 2Current
NCT03380931
2,932 pts·Fabry
2018-062030-08·Recruiting
NCT07528427
506 pts·Fabry
2023-122028-09·Completed
3,438 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-09-102.4y awayPh3 Readout· Fabry
2030-08-094.4y awayPh3 Readout· Fabry
Trial Timeline
Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
P2/3
Recruit…
P2/3
Complet…
Catalysts
Ph3 Readout
2028-09-10 · 2.4y away
Fabry
Ph3 Readout
2030-08-09 · 4.4y away
Fabry
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03380931Phase 2/3FabryRecruiting2932PFS
NCT07528427Phase 2/3FabryCompleted506MRD
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-1085PfizerPreclinicalFXIaPD-L1i
RilulemzoparlimabNovartisPhase 2/3KRASG12DPD-L1i
AZN-6870AstraZenecaPhase 2/3EGFRCDK2i
SNY-9600SanofiNDA/BLAB7-H3PD-L1i
TAK-1836TakedaPreclinicalEGFRKIF18Ai
NirafutibatinibBayerPhase 2WRNPD-L1i
MotainavolisibAmgenNDA/BLACD47PD-L1i
BNT-8090BioNTechPhase 2AuroraAPD-L1i
MiriglumideAlnylamPhase 3CD3PD-L1i
ZanurapivirNeurocrineNDA/BLAEGFRCD47i