← Pipeline|460-4909

460-4909

Preclinical
Source: Trial-derived·Trials: 2
Modality
mRNA
MOA
USP1i
Target
PSMA
Pathway
JAK/STAT
PAHGAEoE
Development Pipeline
Preclinical
Oct 2017
Mar 2026
PreclinicalCurrent
NCT08880726
2,417 pts·EoE
2022-08TBD·Recruiting
NCT05664978
1,034 pts·PAH
2017-102026-03·Recruiting
3,451 total pts2 indications
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-03-162w agoInterim· PAH
Trial Timeline
Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2
Preclinical
Recruit…
Preclinical
Recruit…
Catalysts
Interim
2026-03-16 · 2w ago
PAH
Recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08880726PreclinicalEoERecruiting2417EFS
NCT05664978PreclinicalPAHRecruiting1034Safety
Competitors (10)
DrugCompanyPhaseTargetMOA
AZN-3724AstraZenecaPreclinicalPSMABCMA ADC
DoxacageneSanofiApprovedPSMASHP2i
SNY-2934SanofiPhase 3KRASG12DUSP1i
GSK-2051GSKPhase 1PSMAEGFRi
AMG-9052AmgenPhase 2/3CDK2USP1i
GIL-2445Gilead SciencesPhase 2/3PSMAALKi
DatozumabRegeneronPhase 1B7-H3USP1i
BII-1564BiogenPhase 2PSMABETi
BGN-3859BeiGeneApprovedPSMACD47i
GMA-729GenmabPhase 2BCL-2USP1i