← Pipeline|Lisozanubrutinib

Lisozanubrutinib

NDA/BLA
PST-9459
Source: Trial-derived·Trials: 2
Modality
Fusion Protein
MOA
CDK2i
Target
CD20
Pathway
PI3K/AKT
Cervical CaHeart FailureNSCLC
Development Pipeline
Preclinical
~Jul 2017
~Oct 2018
Phase 1
~Jan 2019
~Apr 2020
Phase 2
~Jul 2020
~Oct 2021
Phase 3
~Jan 2022
~Apr 2023
NDA/BLA
Jul 2023
Apr 2031
NDA/BLACurrent
NCT07474659
2,927 pts·Cervical Ca
2023-072031-04·Completed
NCT04619190
536 pts·Heart Failure
2024-022026-08·Not yet recruiting
3,463 total pts2 indications
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-08-034mo awayPh3 Readout· Heart Failure
2031-04-135.0y awayPh3 Readout· Cervical Ca
Trial Timeline
Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2
NDA/BLA
Complet…
NDA/BLA
Not yet…
Catalysts
Ph3 Readout
2026-08-03 · 4mo away
Heart Failure
Ph3 Readout
2031-04-13 · 5.0y away
Cervical Ca
CompletedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07474659NDA/BLACervical CaCompleted2927OS
NCT04619190NDA/BLAHeart FailureNot yet recr...536NT-proBNP
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-3703PfizerPhase 1/2CDK2CDK2i
JNJ-8637Johnson & JohnsonNDA/BLACD20WEE1i
TirafotisoranRochePhase 2CD38CDK2i
LisolucimabNovartisApprovedCD20KRASG12Ci
ABB-8985AbbViePhase 2CD20MALT1i
ABB-3951AbbViePhase 2/3TNFαCDK2i
AZN-6870AstraZenecaPhase 2/3EGFRCDK2i
TirasotorasibTakedaNDA/BLAIL-17ACDK2i
MavuglumideBayerApprovedGLP-1RCDK2i
DSN-3066Daiichi SankyoPhase 3IL-13CDK2i