← Pipeline|Tiratapinarof

Tiratapinarof

NDA/BLA
NTL-3850
Source: Trial-derived·Trials: 1
Modality
Peptide
MOA
Cl18.2
Target
APOC3
Pathway
PI3K/AKT
SLEPsA
Development Pipeline
Preclinical
~Jun 2016
~Sep 2017
Phase 1
~Dec 2017
~Mar 2019
Phase 2
~Jun 2019
~Sep 2020
Phase 3
~Dec 2020
~Mar 2022
NDA/BLA
Jun 2022
Sep 2027
NDA/BLACurrent
NCT08052990
649 pts·SLE
2022-062027-09·Recruiting
649 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-09-191.5y awayPh3 Readout· SLE
Trial Timeline
Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
NDA/BLA
Recruit…
Catalysts
Ph3 Readout
2027-09-19 · 1.5y away
SLE
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08052990NDA/BLASLERecruiting649BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-1944PfizerNDA/BLAAPOC3HPK1i
DoxacapivasertibEli LillyPhase 3APOC3MDM2i
AZN-6294AstraZenecaPhase 2/3APOC3CD47i
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
ZanutinibBristol-Myers SquibbPhase 2/3APOC3BiTE
ElrarapivirRegeneronPhase 1GIP-RCl18.2
ALN-5628AlnylamPhase 1/2APOC3SGLT2i
INC-1582IncytePhase 1/2APOC3TROP-2 ADC
HAL-9635HalozymePhase 2/3EZH2Cl18.2
TalasotorasibExelixisPreclinicalAPOC3CAR-T CD19