← Pipeline|180-3597

180-3597

Preclinical
Source: Trial-derived·Trials: 2
Modality
Gene Editing
MOA
RAS(ON)i
Target
SHP2
Pathway
Autophagy
Ewing SarcomaLGS
Development Pipeline
Preclinical
Nov 2020
Aug 2030
PreclinicalCurrent
NCT05560121
2,891 pts·Ewing Sarcoma
2020-112030-08·Active
NCT04779591
2,675 pts·LGS
2025-012026-07·Recruiting
5,566 total pts2 indications
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-07-093mo awayInterim· LGS
2030-08-184.4y awayInterim· Ewing Sarcoma
Trial Timeline
Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Preclinical
Active
Preclinical
Recruit…
Catalysts
Interim
2026-07-09 · 3mo away
LGS
Interim
2030-08-18 · 4.4y away
Ewing Sarcoma
RecruitingActive|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05560121PreclinicalEwing SarcomaActive28916MWD
NCT04779591PreclinicalLGSRecruiting2675EASI-75
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-5126NovartisPhase 3SHP2PI3Ki
MRK-1380Merck & CoPreclinicalSHP2SOS1i
MRK-6781Merck & CoApprovedTIGITRAS(ON)i
ABB-1817AbbViePhase 3SHP2WRNi
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
SNY-9073SanofiPhase 2B7-H3RAS(ON)i
TixarelsinVertex PharmaPhase 1ALKRAS(ON)i
MRN-7409ModernaNDA/BLASHP2CDK2i
FixatuximabLegend BiotechPreclinicalCFTRRAS(ON)i