← Pipeline|Bemasotorasib

Bemasotorasib

Phase 2
EXE-1077
Source: Trial-derived·Trials: 2
Modality
Fusion Protein
MOA
IL-23i
Target
CD38
Pathway
DDR
MCLACC
Development Pipeline
Preclinical
~May 2016
~Aug 2017
Phase 1
~Nov 2017
~Feb 2019
Phase 2
May 2019
Jun 2030
Phase 2Current
NCT06820996
685 pts·MCL
2024-092030-06·Recruiting
NCT04185806
2,510 pts·ACC
2019-052028-06·Terminated
3,195 total pts2 indications
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-06-152.2y awayPh2 Data· ACC
2030-06-104.2y awayPh2 Data· MCL
Trial Timeline
Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
P2
Termina…
P2
Recruit…
Catalysts
Ph2 Data
2028-06-15 · 2.2y away
ACC
Ph2 Data
2030-06-10 · 4.2y away
MCL
RecruitingTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06820996Phase 2MCLRecruiting685eGFR
NCT04185806Phase 2ACCTerminated2510FEV1
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
TirafotisoranRochePhase 2CD38CDK2i
NVS-6360NovartisApprovedCD38FXIai
DoxasotorasibAbbViePhase 2CD38VEGFi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
GSK-6983GSKPhase 2ALKIL-23i
MotarapivirGSKPreclinicalAuroraAIL-23i
AMG-2597AmgenPhase 2/3CD38PLK4i
IvosotorasibVertex PharmaPreclinicalCD38BTKi