← Pipeline|Surabrutinib

Surabrutinib

Phase 2
GR-9592
Source: Trial-derived·Trials: 2
Modality
Nanobody
MOA
HPK1i
Target
RET
Pathway
Complement
HCCDLBCL
Development Pipeline
Preclinical
~Sep 2014
~Dec 2015
Phase 1
~Mar 2016
~Jun 2017
Phase 2
Sep 2017
Jul 2027
Phase 2Current
NCT05673682
530 pts·HCC
2017-092026-01·Completed
NCT03398729
242 pts·DLBCL
2021-062027-07·Active
772 total pts2 indications
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-01-212mo agoPh2 Data· HCC
2027-07-101.3y awayPh2 Data· DLBCL
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3
P2
Complet…
P2
Active
Catalysts
Ph2 Data
2026-01-21 · 2mo ago
HCC
Ph2 Data
2027-07-10 · 1.3y away
DLBCL
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05673682Phase 2HCCCompleted530CfB
NCT03398729Phase 2DLBCLActive242VA
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-1944PfizerNDA/BLAAPOC3HPK1i
RHH-5389RochePreclinicalRETSTINGag
NVS-6974NovartisPreclinicalCD19HPK1i
ABB-7516AbbViePhase 3PD-L1HPK1i
FixanesiranAbbViePreclinicalRETJAK1/2i
BMY-8678Bristol-Myers SquibbApprovedRETMDM2i
VRT-1576Vertex PharmaPhase 2/3RETSHP2i
BemanesiranBioNTechPhase 3PLK4HPK1i
BII-5240BiogenPhase 2/3MALT1HPK1i
ARG-3458ArgenxPreclinicalRETIL-17i