← Pipeline|Tezevorutinib

Tezevorutinib

Phase 1/2
512-5678
Source: Trial-derived·Trials: 2
Modality
Vaccine
MOA
PCSK9i
Target
RET
Pathway
JAK/STAT
DravetMDS
Development Pipeline
Preclinical
~Oct 2016
~Jan 2018
Phase 1
Apr 2018
Mar 2029
Phase 1Current
NCT06426455
1,430 pts·Dravet
2018-042029-02·Active
NCT03457682
128 pts·Dravet
2019-122029-03·Terminated
1,558 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-02-092.9y awayPh2 Data· Dravet
2029-03-283.0y awayPh2 Data· Dravet
Trial Timeline
Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2
P1/2
Active
P1/2
Termina…
Catalysts
Ph2 Data
2029-02-09 · 2.9y away
Dravet
Ph2 Data
2029-03-28 · 3.0y away
Dravet
ActiveTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06426455Phase 1/2DravetActive1430PFS
NCT03457682Phase 1/2DravetTerminated128BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
RHH-5389RochePreclinicalRETSTINGag
MRK-8368Merck & CoPhase 3ALKPCSK9i
FixanesiranAbbViePreclinicalRETJAK1/2i
RibofutibatinibAstraZenecaPhase 2/3SOS1PCSK9i
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
BMY-8678Bristol-Myers SquibbApprovedRETMDM2i
PolazasiranAmgenPhase 2LAG-3PCSK9i
CevitinibRegeneronPhase 3FGFRPCSK9i
VRT-1576Vertex PharmaPhase 2/3RETSHP2i
ARG-3458ArgenxPreclinicalRETIL-17i