← Pipeline|Lisotapinarof

Lisotapinarof

NDA/BLA
ABD-646
Source: Trial-derived·Trials: 2
Modality
siRNA
MOA
VEGFi
Target
CD38
Pathway
JAK/STAT
CFNMOSDLN
Development Pipeline
Preclinical
~May 2019
~Aug 2020
Phase 1
~Nov 2020
~Feb 2022
Phase 2
~May 2022
~Aug 2023
Phase 3
~Nov 2023
~Feb 2025
NDA/BLA
May 2025
Aug 2028
NDA/BLACurrent
NCT08065404
1,961 pts·CF
2025-05TBD·Completed
NCT06144255
282 pts·NMOSD
2025-082028-08·Terminated
2,243 total pts2 indications
Approved
CompletedCurrentUpcoming
Catalysts (1)
2028-08-212.4y awayPh3 Readout· NMOSD
Trial Timeline
Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3
NDA/BLA
Complet…
NDA/BLA
Termina…
Catalysts
Ph3 Readout
2028-08-21 · 2.4y away
NMOSD
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08065404NDA/BLACFCompleted1961SRI-4
NCT06144255NDA/BLANMOSDTerminated282EDSS
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
TirafotisoranRochePhase 2CD38CDK2i
NVS-6360NovartisApprovedCD38FXIai
MRK-5413Merck & CoPhase 1GLP-1RVEGFi
DoxasotorasibAbbViePhase 2CD38VEGFi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
CeviderotideNovo NordiskPreclinicalIL-13VEGFi
AMG-2597AmgenPhase 2/3CD38PLK4i
IvosotorasibVertex PharmaPreclinicalCD38BTKi