← Pipeline|Rilusotorasib

Rilusotorasib

Preclinical
PRO-4446
Source: Trial-derived·Trials: 1
Modality
Fusion Protein
MOA
CAR-T BCMA
Target
PLK4
Pathway
Notch
Breast CaEndometrial Ca
Development Pipeline
Preclinical
Nov 2021
Oct 2031
PreclinicalCurrent
NCT05884431
2,089 pts·Endometrial Ca
2021-112031-10·Completed
2,089 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-07-069mo agoBTD· Endometrial Ca
2031-10-115.5y awayInterim· Endometrial Ca
Trial Timeline
Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3Q4
Preclinical
Complet…
Catalysts
BTD
2025-07-06 · 9mo ago
Endometrial Ca
Interim
2031-10-11 · 5.5y away
Endometrial Ca
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05884431PreclinicalEndometrial CaCompleted2089OS
Competitors (10)
DrugCompanyPhaseTargetMOA
VoxacilimabPfizerPhase 2TYK2CAR-T BCMA
NVO-9087Novo NordiskPhase 1/2TauCAR-T BCMA
FixazanubrutinibAmgenPhase 2PI3KαCAR-T BCMA
REG-8074RegeneronPhase 2/3KRASG12CCAR-T BCMA
BemanesiranBioNTechPhase 3PLK4HPK1i
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i
JAZ-8729Jazz PharmaPhase 2/3FcRnCAR-T BCMA
ILM-2412IlluminaPhase 3PLK4AuroraAi