← Pipeline|Tezerelsin

Tezerelsin

Phase 1/2
BLA-7519
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
PLK4i
Target
SOS1
Pathway
Lipid Met
Crohn'sMCC
Development Pipeline
Preclinical
~Jun 2018
~Sep 2019
Phase 1
Dec 2019
Nov 2029
Phase 1Current
NCT05620663
1,635 pts·MCC
2019-122025-05·Completed
NCT03737334
831 pts·Crohn's
2023-102029-11·Active
2,466 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-05-2310mo agoPh2 Data· MCC
2029-11-133.6y awayPh2 Data· Crohn's
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
P1/2
Complet…
P1/2
Active
Catalysts
Ph2 Data
2025-05-23 · 10mo ago
MCC
Ph2 Data
2029-11-13 · 3.6y away
Crohn's
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05620663Phase 1/2MCCCompleted1635PASI75
NCT03737334Phase 1/2Crohn'sActive831Safety
Competitors (10)
DrugCompanyPhaseTargetMOA
TerarelsinAbbViePreclinicalSOS1SOS1i
RibofutibatinibAstraZenecaPhase 2/3SOS1PCSK9i
AMG-2597AmgenPhase 2/3CD38PLK4i
VoxacageneGilead SciencesPhase 2/3SOS1TYK2i
RiluinavolisibModernaNDA/BLAKIF18APLK4i
SRP-9822SareptaPhase 3SOS1FGFRi
FixaosocimabTG TherapeuticsPhase 2/3SOS1PI3Ki
ZanurapivirImmunocorePhase 1SOS1PRMT5i
LiravorutinibBiomea FusionPhase 1/2GPRC5DPLK4i
RilurelsinDynavaxPhase 1/2SOS1BTKi