← Pipeline|Darafutibatinib

Darafutibatinib

Approved
BPT-3277
Source: Trial-derived·Trials: 3
Modality
Nanobody
MOA
HER2
Target
FLT3
Pathway
Complement
ETIgAN
Development Pipeline
Preclinical
~Feb 2012
~May 2013
Phase 1
~Aug 2013
~Nov 2014
Phase 2
~Feb 2015
~May 2016
Phase 3
~Aug 2016
~Nov 2017
NDA/BLA
~Feb 2018
~May 2019
Approved
Aug 2019
Mar 2028
ApprovedCurrent
NCT05664010
430 pts·ET
2025-092025-12·Completed
NCT04240203
2,812 pts·ET
2021-102028-03·Recruiting
NCT08964954
688 pts·IgAN
2019-082027-11·Recruiting
3,930 total pts2 indications
CompletedCurrentUpcoming
Catalysts (3)
2025-12-094mo agoPh3 Readout· ET
2027-11-131.6y awayPh3 Readout· IgAN
2028-03-262.0y awayPh3 Readout· ET
Trial Timeline
Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2
Approved
Recruit…
Approved
Recruit…
Approved
Complet…
Catalysts
Ph3 Readout
2025-12-09 · 4mo ago
ET
Ph3 Readout
2027-11-13 · 1.6y away
IgAN
Ph3 Readout
2028-03-26 · 2.0y away
ET
RecruitingCompleted|StartCompletionToday
Trials (3)
NCTPhaseIndicationStatusNEP
NCT05664010ApprovedETCompleted430ACR20
NCT04240203ApprovedETRecruiting2812CfB
NCT08964954ApprovedIgANRecruiting688ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
JNJ-8168Johnson & JohnsonPhase 2/3FLT3GLP-1/GIP
LLY-8903Eli LillyPreclinicalCD47HER2
SNY-7254SanofiPhase 2CFTRHER2
DatobrutinibSanofiPhase 3HER2
TAK-9344TakedaPhase 3CGRPHER2
SotorapivirModernaApprovedFLT3TYK2i
NidaratamabExelixisPhase 3FLT3AHRant
VoxaderotideViking TherapeuticsApprovedPD-L1HER2
AdagrarapivirIdeaya BioPhase 1/2IL-17AHER2