← Pipeline|Ivosotorasib

Ivosotorasib

Preclinical
VRT-9022
Source: Trial-derived·Trials: 1
Modality
Gene Therapy
MOA
BTKi
Target
CD38
Pathway
Cell Cycle
RSVEwing SarcomaHCC
Development Pipeline
Preclinical
Jul 2017
Nov 2026
PreclinicalCurrent
NCT05969738
2,771 pts·HCC
2017-072026-11·Completed
2,771 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-11-188mo awayInterim· HCC
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q4
Preclinical
Complet…
Catalysts
Interim
2026-11-18 · 8mo away
HCC
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05969738PreclinicalHCCCompleted2771LiverFat
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
TirafotisoranRochePhase 2CD38CDK2i
NVS-6360NovartisApprovedCD38FXIai
DoxasotorasibAbbViePhase 2CD38VEGFi
AZN-8281AstraZenecaPhase 1SHP2BTKi
BMY-3371Bristol-Myers SquibbPhase 3WRNBTKi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
NVO-7872Novo NordiskNDA/BLAB7-H3BTKi
NVO-6275Novo NordiskPhase 1SMN2BTKi