← Pipeline|Terarelsin

Terarelsin

Phase 1/2
ROV-463
Source: Trial-derived·Trials: 2
Modality
Fusion Protein
MOA
Menini
Target
TIGIT
Pathway
Angiogenesis
ADPKDNMOSD
Development Pipeline
Preclinical
~Nov 2017
~Feb 2019
Phase 1
May 2019
Oct 2031
Phase 1Current
NCT04306151
1,139 pts·NMOSD
2019-052031-10·Completed
NCT08390893
1,706 pts·NMOSD
2020-062025-06·Recruiting
2,845 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-06-0810mo agoPh2 Data· NMOSD
2031-10-105.5y awayPh2 Data· NMOSD
Trial Timeline
Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3Q4
P1/2
Complet…
P1/2
Recruit…
Catalysts
Ph2 Data
2025-06-08 · 10mo ago
NMOSD
Ph2 Data
2031-10-10 · 5.5y away
NMOSD
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04306151Phase 1/2NMOSDCompleted1139HAM-D
NCT08390893Phase 1/2NMOSDRecruiting1706BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
ZanuderotideJohnson & JohnsonPhase 2/3TIGITGLP-1/GIP
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
IvorelsinEli LillyApprovedJAK1Menini
MRK-6781Merck & CoApprovedTIGITRAS(ON)i
NVO-2974Novo NordiskNDA/BLAPARPMenini
PexamavacamtenDaiichi SankyoNDA/BLATIGITCD3xCD20
BNT-5232BioNTechNDA/BLATIGITPARPi
ALN-8757AlnylamPreclinicalTIGITCFTRmod
MiritinibNeurocrinePhase 3TIGITSTINGag
UTH-9370United TherapeuticsNDA/BLATIGITPARPi