← Pipeline|Zorinesiran

Zorinesiran

Phase 1/2
TWS-3026
Source: Trial-derived·Trials: 1
Modality
Degrader
MOA
HER2
Target
BCL-2
Pathway
Ferroptosis
IgAN
Development Pipeline
Preclinical
~Aug 2016
~Nov 2017
Phase 1
Feb 2018
Jun 2030
Phase 1Current
NCT03691393
1,999 pts·IgAN
2018-022030-06·Terminated
1,999 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-06-034.2y awayPh2 Data· IgAN
Trial Timeline
2018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
P1/2
Termina…
Catalysts
Ph2 Data
2030-06-03 · 4.2y away
IgAN
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03691393Phase 1/2IgANTerminated1999DAS28
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
LLY-8903Eli LillyPreclinicalCD47HER2
RHH-8550RocheApprovedBCL-2PRMT5i
SNY-7254SanofiPhase 2CFTRHER2
DatobrutinibSanofiPhase 3HER2
TAK-9344TakedaPhase 3CGRPHER2
RimaglumideBiogenPhase 1/2BCL-2IL-17i
ARG-4339ArgenxPhase 2BCL-2TYK2i
GMA-729GenmabPhase 2BCL-2USP1i
HAL-996HalozymePhase 1/2BCL-2BCL-2i