← Pipeline|PCI-3652

PCI-3652

Phase 1
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
MDM2i
Target
IL-23
Pathway
Proteasome
Ovarian CaSchizophreniaHuntington's
Development Pipeline
Preclinical
~Sep 2018
~Dec 2019
Phase 1
Mar 2020
Apr 2030
Phase 1Current
NCT05589701
2,940 pts·Ovarian Ca
2020-032030-04·Not yet recruiting
NCT03532346
2,367 pts·Ovarian Ca
2021-062028-06·Terminated
5,307 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-06-102.2y awayInterim· Ovarian Ca
2030-04-264.1y awayInterim· Ovarian Ca
Trial Timeline
2020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
P1
Not yet…
P1
Termina…
Catalysts
Interim
2028-06-10 · 2.2y away
Ovarian Ca
Interim
2030-04-26 · 4.1y away
Ovarian Ca
TerminatedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05589701Phase 1Ovarian CaNot yet recr...2940PANSS
NCT03532346Phase 1Ovarian CaTerminated2367CfB
Competitors (10)
DrugCompanyPhaseTargetMOA
DoxacapivasertibEli LillyPhase 3APOC3MDM2i
MRK-7739Merck & CoPreclinicalIL-23ALKi
BMY-8678Bristol-Myers SquibbApprovedRETMDM2i
TerasacituzumabNovo NordiskNDA/BLAIL-23KRASG12Ci
DSN-6862Daiichi SankyoPreclinicalIL-23SOS1i
AMG-415AmgenPhase 1CDK2MDM2i
GIL-2037Gilead SciencesApprovedKRASG12DMDM2i
TezecilimabRegeneronApprovedIL-23CGRPant
CapiglumideBioNTechPreclinicalCGRPMDM2i
RimasertibExelixisPhase 3B7-H3MDM2i