← Pipeline|Darasotorasib

Darasotorasib

Preclinical
GUD-4539
Source: Trial-derived·Trials: 1
Modality
ADC
MOA
TNFi
Target
PCSK9
Pathway
STING
ALS
Development Pipeline
Preclinical
Oct 2019
Aug 2029
PreclinicalCurrent
NCT04867737
2,228 pts·ALS
2019-102029-08·Active
2,228 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-08-013.3y awayInterim· ALS
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
Preclinical
Active
Catalysts
Interim
2029-08-01 · 3.3y away
ALS
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04867737PreclinicalALSActive2228DAS28
Competitors (10)
DrugCompanyPhaseTargetMOA
ZanusertibAbbVieApprovedPCSK9KRASG12Di
AZN-7403AstraZenecaPhase 2/3FGFRTNFi
TAK-8262TakedaNDA/BLATauTNFi
TalalemzoparlimabGilead SciencesPhase 1FcRnTNFi
GIL-4361Gilead SciencesPreclinicalPCSK9STINGag
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
RibozanubrutinibGenmabApprovedGPRC5DTNFi
BMR-8377BioMarinPhase 1/2PCSK9BTKi
CapifutibatinibIncytePhase 3PCSK9BCL-2i
INC-5849IncytePhase 2PCSK9STINGag