← Pipeline|GEN-516

GEN-516

Phase 2/3
Source: Trial-derived·Trials: 1
Modality
mRNA
MOA
VEGFi
Target
PLK4
Pathway
PI3K/AKT
NBHCC
Development Pipeline
Preclinical
~Dec 2016
~Mar 2018
Phase 1
~Jun 2018
~Sep 2019
Phase 2
Dec 2019
Jul 2026
Phase 2Current
NCT07632868
1,288 pts·NB
2019-122026-07·Terminated
1,288 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-07-013mo awayPh3 Readout· NB
Trial Timeline
2020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3
P2/3
Termina…
Catalysts
Ph3 Readout
2026-07-01 · 3mo away
NB
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07632868Phase 2/3NBTerminated1288PANSS
Competitors (10)
DrugCompanyPhaseTargetMOA
MRK-5413Merck & CoPhase 1GLP-1RVEGFi
DoxasotorasibAbbViePhase 2CD38VEGFi
CeviderotideNovo NordiskPreclinicalIL-13VEGFi
VRT-6833Vertex PharmaPreclinicalALKVEGFi
BemanesiranBioNTechPhase 3PLK4HPK1i
BGN-8936BeiGenePhase 1/2FXIaVEGFi
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
CapifutibatinibIntra-CellularPhase 3GIP-RVEGFi
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i