← Pipeline|Pexavorutinib

Pexavorutinib

Preclinical
DAI-8075
Source: Trial-derived·Trials: 1
Modality
Multispecific
MOA
TROP-2 ADC
Target
GIP-R
Pathway
Amyloid
MCL
Development Pipeline
Preclinical
Aug 2021
Nov 2026
PreclinicalCurrent
NCT05070703
146 pts·MCL
2021-082026-11·Recruiting
146 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-11-027mo awayInterim· MCL
Trial Timeline
Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q4
Preclinical
Recruit…
Catalysts
Interim
2026-11-02 · 7mo away
MCL
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05070703PreclinicalMCLRecruiting146ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-5094Johnson & JohnsonPhase 2/3GIP-REGFRi
RHH-3592RochePhase 1/2GIP-RBCL-2i
AZN-5978AstraZenecaPhase 2/3GIP-RAHRant
IvotuximabGSKNDA/BLAGIP-RKRASG12Di
BAY-6520BayerPhase 2AHRTROP-2 ADC
BemazumabRegeneronPhase 1VEGFTROP-2 ADC
ElrarapivirRegeneronPhase 1GIP-RCl18.2
GMA-5010GenmabPhase 3JAK2TROP-2 ADC
INC-1582IncytePhase 1/2APOC3TROP-2 ADC
CapifutibatinibIntra-CellularPhase 3GIP-RVEGFi