← Pipeline|Terafutibatinib

Terafutibatinib

Phase 2/3
RET-9812
Source: Trial-derived·Trials: 2
Modality
Gene Editing
MOA
Anti-Aβ
Target
TYK2
Pathway
Epigenetic
PAH
Development Pipeline
Preclinical
~Mar 2021
~Jun 2022
Phase 1
~Sep 2022
~Dec 2023
Phase 2
Mar 2024
Jun 2027
Phase 2Current
NCT03987606
1,839 pts·PAH
2024-03TBD·Recruiting
NCT07336027
451 pts·PAH
2025-042027-06·Completed
2,290 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-06-251.2y awayPh3 Readout· PAH
Trial Timeline
Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3
P2/3
Recruit…
P2/3
Complet…
Catalysts
Ph3 Readout
2027-06-25 · 1.2y away
PAH
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03987606Phase 2/3PAHRecruiting1839DOR
NCT07336027Phase 2/3PAHCompleted451BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
VoxacilimabPfizerPhase 2TYK2CAR-T BCMA
LLY-8369Eli LillyApprovedMeninAnti-Aβ
MRK-3732Merck & CoPhase 1TYK2PARPi
ABB-8696AbbViePhase 3BCMAAnti-Aβ
BAY-6035BayerPhase 1C5Anti-Aβ
ZenotinibBioNTechPhase 1CGRPAnti-Aβ
COR-9566CorceptApprovedTYK2HPK1i
RLA-6817Relay TherapeuticsPhase 3TIGITAnti-Aβ
LisoosocimabZealand PharmaApprovedKIF18AAnti-Aβ
PRA-419Praxis PrecisionApprovedCl18.2Anti-Aβ