← Pipeline|Bemasertib

Bemasertib

Phase 1
ACH-3903
Source: Trial-derived·Trials: 2
Modality
mRNA
MOA
GLP-1ag
Target
PLK4
Pathway
Tau
DravetCholangiocarcinomaNSCLC
Development Pipeline
Preclinical
~Dec 2023
~Mar 2025
Phase 1
Jun 2025
Mar 2030
Phase 1Current
NCT04053110
1,543 pts·NSCLC
2025-072030-03·Active
NCT03741438
949 pts·NSCLC
2025-062029-11·Completed
2,492 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-11-063.6y awayInterim· NSCLC
2030-03-154.0y awayInterim· NSCLC
Trial Timeline
Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
P1
Complet…
P1
Active
Catalysts
Interim
2029-11-06 · 3.6y away
NSCLC
Interim
2030-03-15 · 4.0y away
NSCLC
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04053110Phase 1NSCLCActive1543CR
NCT03741438Phase 1NSCLCCompleted949OS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-8662PfizerNDA/BLACD19GLP-1ag
NVO-7840Novo NordiskPhase 2/3B7-H3GLP-1ag
MRN-7601ModernaPhase 2IL-13GLP-1ag
BemanesiranBioNTechPhase 3PLK4HPK1i
ARG-1250ArgenxPhase 2C5GLP-1ag
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i
ILM-5680IlluminaPhase 2BETGLP-1ag
ILM-2412IlluminaPhase 3PLK4AuroraAi