← Pipeline|Doxafutibatinib

Doxafutibatinib

Phase 1
PMN-8834
Source: Trial-derived·Trials: 1
Modality
siRNA
MOA
PCSK9i
Target
MDM2
Pathway
Wnt
MG
Development Pipeline
Preclinical
~Jan 2019
~Apr 2020
Phase 1
Jul 2020
May 2030
Phase 1Current
NCT05714419
1,678 pts·MG
2020-072030-05·Completed
1,678 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-05-044.1y awayInterim· MG
Trial Timeline
Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
P1
Complet…
Catalysts
Interim
2030-05-04 · 4.1y away
MG
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05714419Phase 1MGCompleted1678UPCR
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-6079Eli LillyPhase 2MDM2PRMT5i
LLY-3251Eli LillyPhase 2MDM2BiTE
MRK-8368Merck & CoPhase 3ALKPCSK9i
RibofutibatinibAstraZenecaPhase 2/3SOS1PCSK9i
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
GSK-7987GSKPhase 3MDM2PD-1i
PolazasiranAmgenPhase 2LAG-3PCSK9i
AMG-2752AmgenPreclinicalMDM2WRNi
REG-3155RegeneronPhase 1/2MDM2PI3Ki
CevitinibRegeneronPhase 3FGFRPCSK9i