← Pipeline|Zorivorutinib

Zorivorutinib

Approved
BMY-6101
Source: Trial-derived·Trials: 4
Modality
mRNA
MOA
Cl18.2
Target
DLL3
Pathway
Lipid Met
Prostate CaMMT2D
Development Pipeline
Preclinical
~Apr 2011
~Jul 2012
Phase 1
~Oct 2012
~Jan 2014
Phase 2
~Apr 2014
~Jul 2015
Phase 3
~Oct 2015
~Jan 2017
NDA/BLA
~Apr 2017
~Jul 2018
Approved
Oct 2018
Sep 2029
ApprovedCurrent
NCT05160918
525 pts·Prostate Ca
2022-042025-01·Terminated
NCT06737708
1,353 pts·T2D
2018-102026-06·Completed
NCT04555539
2,934 pts·Prostate Ca
2023-112029-09·Terminated
+1 more trial
6,370 total pts3 indications
CompletedCurrentUpcoming
Catalysts (4)
2025-01-081.2y agoPh3 Readout· Prostate Ca
2026-06-163mo awayPh3 Readout· T2D
2026-06-213mo awayPh3 Readout· MM
2029-09-263.5y awayPh3 Readout· Prostate Ca
Trial Timeline
Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
Approved
Complet…
Approved
Termina…
Approved
Not yet…
Approved
Termina…
Catalysts
Ph3 Readout
2025-01-08 · 1.2y ago
Prostate Ca
Ph3 Readout
2026-06-16 · 3mo away
T2D
Ph3 Readout
2026-06-21 · 3mo away
MM
Ph3 Readout
2029-09-26 · 3.5y away
Prostate Ca
CompletedTerminatedNot yet recruiting|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT05160918ApprovedProstate CaTerminated5256MWD
NCT06737708ApprovedT2DCompleted1353MRD
NCT04555539ApprovedProstate CaTerminated2934UPCR
NCT07664985ApprovedMMNot yet recr...1558PFS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
ZenonesiranGSKPreclinicalDLL3CD47i
AMG-7379AmgenPreclinicalDLL3CD47i
ElrarapivirRegeneronPhase 1GIP-RCl18.2
ARG-1924ArgenxPreclinicalDLL3JAK1i
CevinaritideGenmabPhase 2/3DLL3PD-1i
HAL-9635HalozymePhase 2/3EZH2Cl18.2
VKT-6548Viking TherapeuticsPhase 2/3PD-L1Cl18.2
TiratapinarofIntelliaNDA/BLAAPOC3Cl18.2