← Pipeline|Motarasimod

Motarasimod

Phase 2
REP-7974
Source: Trial-derived·Trials: 2
Modality
mAb
MOA
GLP-1ag
Target
PCSK9
Pathway
Cell Cycle
MGBreast CaRB
Development Pipeline
Preclinical
~Dec 2015
~Mar 2017
Phase 1
~Jun 2017
~Sep 2018
Phase 2
Dec 2018
Feb 2025
Phase 2Current
NCT07724786
1,343 pts·RB
2019-032025-02·Recruiting
NCT04798432
2,409 pts·RB
2018-12TBD·Recruiting
3,752 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-02-071.1y agoPh2 Data· RB
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025
P2
Recruit…
P2
Recruit…
Catalysts
Ph2 Data
2025-02-07 · 1.1y ago
RB
Recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07724786Phase 2RBRecruiting1343HAM-D
NCT04798432Phase 2RBRecruiting2409NT-proBNP
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-8662PfizerNDA/BLACD19GLP-1ag
ZanusertibAbbVieApprovedPCSK9KRASG12Di
NVO-7840Novo NordiskPhase 2/3B7-H3GLP-1ag
GIL-4361Gilead SciencesPreclinicalPCSK9STINGag
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
MRN-7601ModernaPhase 2IL-13GLP-1ag
ARG-1250ArgenxPhase 2C5GLP-1ag
BMR-8377BioMarinPhase 1/2PCSK9BTKi
CapifutibatinibIncytePhase 3PCSK9BCL-2i
INC-5849IncytePhase 2PCSK9STINGag