← Pipeline|Pexasotorasib

Pexasotorasib

Phase 1
OMG-5970
Source: Trial-derived·Trials: 2
Modality
Small Molecule
MOA
PD-1i
Target
IL-13
Pathway
Innate Imm
WilmsMDS
Development Pipeline
Preclinical
~Jan 2020
~Apr 2021
Phase 1
Jul 2021
Jul 2029
Phase 1Current
NCT04994874
1,375 pts·MDS
2024-102026-05·Active
NCT05750723
2,901 pts·Wilms
2021-072029-07·Not yet recruiting
4,276 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-05-222mo awayInterim· MDS
2029-07-033.3y awayInterim· Wilms
Trial Timeline
Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
P1
Not yet…
P1
Active
Catalysts
Interim
2026-05-22 · 2mo away
MDS
Interim
2029-07-03 · 3.3y away
Wilms
ActiveNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04994874Phase 1MDSActive1375Biomarker
NCT05750723Phase 1WilmsNot yet recr...2901ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
LisonaritideEli LillyPhase 3IL-13TYK2i
SovarapivirAbbViePhase 2/3IL-13BETi
CeviderotideNovo NordiskPreclinicalIL-13VEGFi
GSK-7987GSKPhase 3MDM2PD-1i
DSN-3066Daiichi SankyoPhase 3IL-13CDK2i
MRN-7601ModernaPhase 2IL-13GLP-1ag
NirabrutinibBioNTechPhase 2/3CDK2PD-1i
CevinaritideGenmabPhase 2/3DLL3PD-1i
ElrarapivirIovancePhase 2IL-13BCL-2i
ZYM-2450ZymeworksPhase 2GLP-1RPD-1i