← Pipeline|Elrazanubrutinib

Elrazanubrutinib

NDA/BLA
CRV-763
Source: Trial-derived·Trials: 2
Modality
Gene Therapy
MOA
GLP-1ag
Target
PLK4
Pathway
Proteasome
PAH
Development Pipeline
Preclinical
~Nov 2017
~Feb 2019
Phase 1
~May 2019
~Aug 2020
Phase 2
~Nov 2020
~Feb 2022
Phase 3
~May 2022
~Aug 2023
NDA/BLA
Nov 2023
Jul 2028
NDA/BLACurrent
NCT03410549
2,302 pts·PAH
2025-062026-02·Active
NCT07565348
146 pts·PAH
2023-112028-07·Terminated
2,448 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-02-072mo agoPh3 Readout· PAH
2028-07-132.3y awayPh3 Readout· PAH
Trial Timeline
Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3
NDA/BLA
Termina…
NDA/BLA
Active
Catalysts
Ph3 Readout
2026-02-07 · 2mo ago
PAH
Ph3 Readout
2028-07-13 · 2.3y away
PAH
ActiveTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03410549NDA/BLAPAHActive2302CfB
NCT07565348NDA/BLAPAHTerminated146PFS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-8662PfizerNDA/BLACD19GLP-1ag
NVO-7840Novo NordiskPhase 2/3B7-H3GLP-1ag
MRN-7601ModernaPhase 2IL-13GLP-1ag
BemanesiranBioNTechPhase 3PLK4HPK1i
ARG-1250ArgenxPhase 2C5GLP-1ag
PeminaritideSareptaNDA/BLAPLK4JAK1/2i
PexaosocimabUnited TherapeuticsNDA/BLAPLK4KRASG12Ci
PolalucimabJazz PharmaPreclinicalPLK4EZH2i
ILM-5680IlluminaPhase 2BETGLP-1ag
ILM-2412IlluminaPhase 3PLK4AuroraAi