← Pipeline|Zorisotorasib

Zorisotorasib

Phase 1
AZN-2601
Source: Trial-derived·Trials: 1
Modality
Cell Therapy
MOA
TYK2i
Target
WRN
Pathway
Notch
PAHT2DMM
Development Pipeline
Preclinical
~Aug 2016
~Nov 2017
Phase 1
Feb 2018
Sep 2029
Phase 1Current
NCT04699747
1,984 pts·PAH
2018-022029-09·Terminated
1,984 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-09-133.5y awayInterim· PAH
Trial Timeline
2018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
P1
Termina…
Catalysts
Interim
2029-09-13 · 3.5y away
PAH
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04699747Phase 1PAHTerminated1984UPCR
Competitors (10)
DrugCompanyPhaseTargetMOA
NidasacituzumabEli LillyApprovedCFTRTYK2i
LisonaritideEli LillyPhase 3IL-13TYK2i
MRK-3745Merck & CoPhase 2WRNFXIai
MRK-2473Merck & CoPhase 1/2Nectin-4TYK2i
BMY-3371Bristol-Myers SquibbPhase 3WRNBTKi
SNY-8628SanofiNDA/BLAB7-H3TYK2i
LisorapivirTakedaPreclinicalWRNBTKi
NirafutibatinibBayerPhase 2WRNPD-L1i
VoxacageneGilead SciencesPhase 2/3SOS1TYK2i
SotosacituzumabVertex PharmaPhase 1METTYK2i