← Pipeline|Terafutibatinib

Terafutibatinib

Phase 1/2
PFE-3646
Source: Trial-derived·Trials: 2
Modality
ASO
MOA
CGRPant
Target
CD38
Pathway
NF-κB
CeliacGastric Ca
Development Pipeline
Preclinical
~Feb 2019
~May 2020
Phase 1
Aug 2020
Apr 2026
Phase 1Current
NCT05275202
742 pts·Celiac
2023-06TBD·Recruiting
NCT08559699
2,677 pts·Gastric Ca
2020-082026-04·Not yet recruiting
3,419 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-04-01tomorrowPh2 Data· Gastric Ca
Trial Timeline
Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2
P1/2
Not yet…
P1/2
Recruit…
Catalysts
Ph2 Data
2026-04-01 · tomorrow
Gastric Ca
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05275202Phase 1/2CeliacRecruiting742VA
NCT08559699Phase 1/2Gastric CaNot yet recr...2677PFS
Competitors (10)
DrugCompanyPhaseTargetMOA
SotovorutinibPfizerApprovedCGRPant
TirafotisoranRochePhase 2CD38CDK2i
NVS-6360NovartisApprovedCD38FXIai
ABB-3060AbbViePhase 2LAG-3CGRPant
DoxasotorasibAbbViePhase 2CD38VEGFi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
AMG-2597AmgenPhase 2/3CD38PLK4i
GIL-6239Gilead SciencesPhase 2TNFαCGRPant
TezecilimabRegeneronApprovedIL-23CGRPant