← Pipeline|Zoribrutinib

Zoribrutinib

Phase 1/2
PRO-6769
Source: Trial-derived·Trials: 1
Modality
Multispecific
MOA
HER2
Target
DLL3
Pathway
mTOR
MCLMigraine
Development Pipeline
Preclinical
~Jan 2020
~Apr 2021
Phase 1
Jul 2021
Apr 2026
Phase 1Current
NCT04593283
1,362 pts·MCL
2021-072026-04·Not yet recruiting
1,362 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-04-243w awayPh2 Data· MCL
Trial Timeline
Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2
P1/2
Not yet…
Catalysts
Ph2 Data
2026-04-24 · 3w away
MCL
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04593283Phase 1/2MCLNot yet recr...1362DOR
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
LLY-8903Eli LillyPreclinicalCD47HER2
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
SNY-7254SanofiPhase 2CFTRHER2
DatobrutinibSanofiPhase 3HER2
ZenonesiranGSKPreclinicalDLL3CD47i
TAK-9344TakedaPhase 3CGRPHER2
AMG-7379AmgenPreclinicalDLL3CD47i
ARG-1924ArgenxPreclinicalDLL3JAK1i