← Pipeline|Pexazanubrutinib

Pexazanubrutinib

Phase 1/2
PHA-9801
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
Anti-Tau
Target
BTK
Pathway
DDR
PNHPancreatic Ca
Development Pipeline
Preclinical
~May 2016
~Aug 2017
Phase 1
Nov 2017
Jul 2029
Phase 1Current
NCT06664532
349 pts·Pancreatic Ca
2017-112029-01·Terminated
NCT03972054
2,320 pts·Pancreatic Ca
2021-062029-07·Completed
2,669 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-01-112.8y awayPh2 Data· Pancreatic Ca
2029-07-183.3y awayPh2 Data· Pancreatic Ca
Trial Timeline
Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
P1/2
Termina…
P1/2
Complet…
Catalysts
Ph2 Data
2029-01-11 · 2.8y away
Pancreatic Ca
Ph2 Data
2029-07-18 · 3.3y away
Pancreatic Ca
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06664532Phase 1/2Pancreatic CaTerminated349UPCR
NCT03972054Phase 1/2Pancreatic CaCompleted2320ORR
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5501PfizerPhase 1BTKBCL-2i
RHH-7558RochePhase 1SGLT2Anti-Tau
RHH-8482RochePhase 1BTKKIF18Ai
NVS-5439NovartisPreclinicalBETAnti-Tau
NVO-9630Novo NordiskPhase 2CD3Anti-Tau
ZorizanubrutinibNovo NordiskPhase 1BTKCD3xCD20
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
BGN-3305BeiGenePhase 2BCMAAnti-Tau
SovarasimodHalozymePhase 1/2WEE1Anti-Tau
369-8021Hansoh PharmaApprovedBTKBETi