← Pipeline|MRK-1380

MRK-1380

Preclinical
Source: Trial-derived·Trials: 2
Modality
Peptide
MOA
SOS1i
Target
SHP2
Pathway
JAK/STAT
Prostate Ca
Development Pipeline
Preclinical
Jan 2022
Mar 2027
PreclinicalCurrent
NCT04412401
664 pts·Prostate Ca
2022-02TBD·Completed
NCT08172774
785 pts·Prostate Ca
2022-012027-03·Completed
1,449 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-03-1611mo awayInterim· Prostate Ca
Trial Timeline
2022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2
Preclinical
Complet…
Preclinical
Complet…
Catalysts
Interim
2027-03-16 · 11mo away
Prostate Ca
Completed|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04412401PreclinicalProstate CaCompleted664SeizFreq
NCT08172774PreclinicalProstate CaCompleted785OS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-2901PfizerPhase 2AHRSOS1i
NVS-5126NovartisPhase 3SHP2PI3Ki
ABB-1817AbbViePhase 3SHP2WRNi
TerarelsinAbbViePreclinicalSOS1SOS1i
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
DoxarapivirBristol-Myers SquibbPhase 3KRASG12CSOS1i
DSN-6862Daiichi SankyoPreclinicalIL-23SOS1i
GIL-2011Gilead SciencesPreclinicalVEGFSOS1i
REG-647RegeneronPreclinicalSMN2SOS1i